Understanding anaesthetics: Ethanol partitioning into lipid membranes, effects on fluidity and permeability

DOI

Ethanol plays an important role in the human metabolism. It is in particular known to act as a drug enhancer by increasing trans-membrane permeability, and as an anesthetic. However, the molecular mechanism behind these functionalities remains largely unknown. In this combined proposal we propose to study molecular structure and dynamics of a lipid membrane containing ethanol. Position and partitioning of ethanol and water molecules will be determined from reflectivity measurements using OFFSPEC. In-plane and trans-membrane dynamics will be determined using the unique capabilities of LET. By using solid supported, highly oriented membranes, we will be able to measure in-plane and trans-membrane diffusive and transport dynamics in-situ, under physiological conditions. Deuterium labeling will be used to emphasize ethanol, water and lipid molecules.

Identifier
DOI https://doi.org/10.5286/ISIS.E.24091189
Metadata Access https://icatisis.esc.rl.ac.uk/oaipmh/request?verb=GetRecord&metadataPrefix=oai_datacite&identifier=oai:icatisis.esc.rl.ac.uk:inv/24091189
Provenance
Creator Dr Victoria Garcia Sakai; Professor Maikel Rheinstadter; Ms Laura Toppozini
Publisher ISIS Neutron and Muon Source
Publication Year 2016
Rights CC-BY Attribution 4.0 International; https://creativecommons.org/licenses/by/4.0/
OpenAccess true
Contact isisdata(at)stfc.ac.uk
Representation
Resource Type Dataset
Discipline Photon- and Neutron Geosciences
Temporal Coverage Begin 2013-07-31T07:12:16Z
Temporal Coverage End 2013-08-29T09:29:13Z